供货周期: | 一周 |
品牌: | 爱必信 |
规格: | 99% |
货号: | abs815976 |
CAS号: | 552-41-0 |
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抑制剂描述: 产品名称:Paeonol 产品别名:见爱必信官网 英文别名:Paeonol 靶点:Phenols CAS:552-41-0 纯度:99% 外观:见爱必信官网 保存方法:store at -20℃ for one year(Powder); in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months. 描述: Paeonol (Peonol), a phenolic compound extracted from Chinese herbs Paeonia suffruticosa (moutan cortex) and Cynanchum paniculatum, inhibits MAO with an IC50 of about 50 μM. 溶解性:Ethanol : 33 mg/mL (198.59 mM) 体外研究: Paeonol is found to be inhibitory against MAO A in a dose-dependent manner with IC50 value of 54.6 μM. Paeonol is shown to inhibit MAO-B in a dose-dependent manner with the IC50 of 42.5 μM. For Paeonol, the Ki is estimated to be 51.1 μM. The inhibition of Paeonol on MAO B is of competitive type with Ki value of 38.2 μM. 体内研究:The 200 mg/kg Paeonol+I/R group .
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