参考价: ¥ 887
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  • 型号:
  • 供货周期:
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抑制剂描述:

产品名称:4-Hydroxytamoxifen

产品别名:见爱必信官网

英文别名:4-Hydroxytamoxifen

靶点:Others

CAS:68392-35-8

纯度:99.18 %

外观:见爱必信官网

保存方法:store at -20℃ for one year(Powder); in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months.

描述:4-Hydroxytamoxifen is the active metabolite of tamoxifen and a selective <b>estrogen receptor (ER)</b> modulator that is widely used in the therapeutic and chemopreventive treatment of breast cancer.

溶解性:体外:
DMSO 77mg/mL(198.7mM)
Water <1mg/mL
Ethanol <1mg/mL

体外研究:

4-OHT is a potent activator of ER and has been shown to have a higher affinity for estrogen receptors compared to tamoxifen. It has significant dose and time-dependent direct effects to alter the contractile function of isolated adult rat cardiac myocytes. 4-HT activates on-target modification frequency for intein-Cas9 variants .

体内研究:

产品信息订购:

  产品货号   产品名称   规格 价格 大包装及货期
  abs816150   4-Hydroxytamoxifen   10mg   887.00   立即咨询
  abs816150   4-Hydroxytamoxifen   50mg   3460.00   立即咨询

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