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抑制剂描述: 产品名称:4-Hydroxytamoxifen 产品别名:见爱必信官网 英文别名:4-Hydroxytamoxifen 靶点:Others CAS:68392-35-8 纯度:99.18 % 外观:见爱必信官网 保存方法:store at -20℃ for one year(Powder); in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months. 描述:4-Hydroxytamoxifen is the active metabolite of tamoxifen and a selective <b>estrogen receptor (ER)</b> modulator that is widely used in the therapeutic and chemopreventive treatment of breast cancer. 溶解性:体外: 体外研究: 4-OHT is a potent activator of ER and has been shown to have a higher affinity for estrogen receptors compared to tamoxifen. It has significant dose and time-dependent direct effects to alter the contractile function of isolated adult rat cardiac myocytes. 4-HT activates on-target modification frequency for intein-Cas9 variants . 体内研究:
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