【序号】:1 【作者】:Thomas H. Marsilje , Wei Pei , Bei Chen , Wenshuo Lu , ,,, 【题名】:Synthesis, Structure–Activity Relationships, and in Vivo Efficacy of the Novel Potent and Selective Anaplastic Lymphoma Kinase (ALK) Inhibitor 5-Chloro-N2-(2-isopropoxy-5-methyl-4-(piperidin-4-yl)phenyl)-N4-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine (LDK378) Currently in Phase 1 and Phase 2 Clinical Trials 【期刊】:J. Med. Chem. 【年、卷、期、起止页码】:J. Med. Chem., 2013, 56 (14), pp 5675–5690 【全文链接】:http://pubs.acs.org/doi/abs/10.1021/jm400402q