供货周期: | 7天 |
品牌: | 爱必信 |
型号: | 99% |
货号: | abs817858 |
CAS号: | 345630-40-2 |
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抑制剂描述: 产品名称:SF1670 产品别名:见爱必信官网 英文别名:SF1670 靶点:PTEN CAS:345630-40-2 纯度:99% 外观:见爱必信官网 保存方法:store at -20℃ for one year(Powder); in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months. 描述: SF1670是一种高度有效且专一的PTEN的抑制剂,其IC50 为 2 μM。 溶解性:DMSO :30.7 mg/mL (100 mM) 体外研究: SF1670 shows potent cytotoxicity in HBEC, PC-3, H1299 cells with IC50 of 5 μM, 10 μM, 44 μM, respectively. In a mouse aortic ring matrigel angiogenesis model, SF1670 stimulates the angiogenic processes. SF1670 augments chemoattractant-elicited PtdIns(3,4,5)P3 signaling in neutrophils and enhances neutrophil functions. 体内研究:Pretreatment of SF1670 (500 nM i.v.) augments bacteria-killing capability in neutropenic mice in both peritonitis and bacterial pneumonia, and decreases the mortality of neutropenia-related pneumonia.
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