供货周期: | 一周 |
品牌: | 爱必信 |
规格: | 98% |
货号: | abs821085 |
CAS号: | 1642288-47-8 |
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抑制剂描述: 产品名称:Mavacamten 产品别名:见爱必信官网 英文别名:Mavacamten 靶点:Myosin CAS:1642288-47-8 纯度:98% 外观:见爱必信官网 保存方法:store at -20℃ for one year(Powder) 描述:Mavacamten is a modulator of cardiac myosin, with IC50s of 490, 711 nM for bovine cardiac and human cardiac, respectively. 溶解性: 体外研究: Mavacamten is found to have an IC50 value of 490 nM in the bovine system, 711 nM in the human system, and 2140 nM in the rabbit system, indicating selectivity of >4-fold for cardiac myosin. 体内研究:Mavacamten is found to have an IC50 value of 490 nM in the bovine system, 711 nM in the human system, and 2140 nM in the rabbit system, indicating selectivity of >4-fold for cardiac myosin.
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