| 供货周期： | 一周 |
| 品牌： | 爱必信 |
| 规格： | >98% |
| 货号： | abs813962 |
| CAS号： | 871224-64-5 |
| 公告提醒：爱必信所有产品和服务仅用于科学研究，不用于临床应用及其他用途提供产品和服务（也不为任何个人提供产品和服务）!
抑制剂描述： 产品名称：Almorexant 产品别名：见爱必信官网 英文别名：Almorexant 靶点：OX Receptor CAS：871224-64-5 纯度：>98% 外观：见爱必信官网 保存方法：store at -20℃ for one year（Powder）； in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months. 描述： Almorexant (ACT-078573) is a competitive OX1 and OX2 orexin receptor antagonist with IC50 of 13 and 8 nM, respectively. It is rapidly absorbed and distributed and shows no tendency to accumulate with repeated dosing. Preclinical studies in rats and dogs have demonstrated a sleep-promoting effect which resembles physiological sleep; this could be quickly reversed upon sensorimotor stimulation and yet allow resumption of sleep upon its cessation. Almorexant’s (ACT-078573) sleep-promoting effects were confirmed in volunteers and patients with primary insomnia. It dose-dependently increased sleep efficiency and decreased sleep latency and wake time after sleep onset. 溶解性：DMSO : ≥ 46 mg/mL 体外研究： 体内研究：
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