Quinidine sulfate dihydrate

Quinidine sulfate dihydrate

参考价:¥1365
供货周期: 一周
品牌: 爱必信
规格: 98%
货号: abs814921
CAS号: 6591-63-5
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抑制剂描述:

产品名称:Quinidine sulfate dihydrate

产品别名:见爱必信官网

英文别名:Quinidine sulfate dihydrate

靶点:Sodium Channel

CAS:6591-63-5

纯度:98%

外观:见爱必信官网

保存方法:Store at -20° C

描述:

Quinidine sulfate dihydrate is a diastereomer of quinine and a Na+ channel blocker. Also a class I antiarrhythmic drug.

溶解性:

体外研究:

Quinidine selectively reduces the proliferation of merlin-deficient HMM cell lines by causing a G0/G1 arrest, whereas the proliferation rates of merlinexpressing HMM cell lines remain unchanged. In addtion to its function as a channel blocker, quinidine is an inhibitor of a specific isoform of the cytochrome P450 family (CYP2D6), which is involved in the detoxification and metabolism of multiple commonly prescribed drugs as well as numerous endogenous substrates.

体内研究:Quinidine is a potent and selective inhibitor of P450db and that quinidine can inhibit the in vivo metabolism of debrisoquine in humans. Quinidine is an inhibitor of amphetamine metabolism in vivo.

产品信息订购:

  产品货号   产品名称   规格 价格 大包装及货期
  abs814921   Quinidine sulfate dihydrate   5g   1365.00   立即咨询
  abs814921   Quinidine sulfate dihydrate   1g   368.00   立即咨询

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