供货周期: | 一周 |
品牌: | 爱必信 |
规格: | |
货号: | abs821180 |
CAS号: | 177469-96-4 |
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抑制剂描述: 产品名称:Implitapide 产品别名:见爱必信官网 英文别名:Implitapide 靶点:MTP CAS:177469-96-4 纯度: 外观:见爱必信官网 保存方法:store at -20℃ for one year(Powder) 描述:Implitapide (AEGR 427) is a microsomal triglyceride transfer protein (MTP) inhibitor. 溶解性:10 mM in DMSO 体外研究: Implitapide suppresses MTP activity using a recombinant human form complexed with protein disulphide isomerase (IC50=10 nM) and inhibit secretion of apoB-containing very low-density lipoprotein (VLDL)-like lipoproteins from a human hepatoma cell (HepG2) with an IC50 value of 1.1 nM. 体内研究:Implitapide suppresses MTP activity using a recombinant human form complexed with protein disulphide isomerase (IC50=10 nM) and inhibit secretion of apoB-containing very low-density lipoprotein (VLDL)-like lipoproteins from a human hepatoma cell (HepG2) with an IC50 value of 1.1 nM.
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