供货周期: | 现货 |
品牌: | 爱必信 |
规格: | 1mg |
货号: | abs9107 |
CAS号: | 16561-29-8 |
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试剂描述: 产品名称:PMA,佛波酯 产品别名:佛波醇12-十四酸酯13-乙酸酯(佛波酯);12-十四酸酯13-乙酸佛波醇酯;Phorbol-12-Myristate-13-Acetate;12-O-tetradecanoyl phorbol-13-acetate CAS号:16561-29-8 英文别名:PMA 分子量:616.83 分子式:C36H56O8 纯度:≥98% 外观:见爱必信官网 保存方法:Store at -20° C,3 years. 描述: PMA (Phorbol-12-Myristate-13-Acetate) is a diester of phorbol and is a tumor promoting compound extracted from croton oil. It is a reversible, highly potent protein kinase C (PKC) activator in vitro and in vivo at nM concentrations. PMA’s effects on PKC are attributed to its similarity to diacylgylerol, a natural activator of PKC. PMA activates Ca2+-ATPase and potentiates forskolin-induced cAMP formation. It has been shown to inhibit apoptosis induced by the Fas antigen, but PMA induces apoptosis in HL-60 promyelocytic leukemia cells. PMA(同义名:TPA)是一种广泛用于体内外实验的佛波酯(phorbol ester) PKC激活剂。PMA结合PKC(Ki =2.6 nM)并激活其功能,在细胞和组织中都呈现出极其广的抑制谱。PMA可以抑制Fas诱导的细胞凋亡,但又可以诱导HL-60细胞的凋亡。PMA是一种高效的肿瘤促进剂,可以促进小鼠皮肤瘤的形成。尽管PMA毒性较强,但是在人体内仍显示出抗白血病和抗中性白细胞减少的活性。 应用:A reversible and highly potent protein kinase C (PKC) activator |
产品信息订购:
产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 |
abs9107 | PMA | 1mg | 560.00 | 立即咨询 |
abs9107 | PMA | 5mg | 1317.00 | 立即咨询 |
abs9107 | PMA | 25mg | 3950.00 | 立即咨询 |
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