【序号】:1 【作者】:Okada H1, Inoue Y, Heya T, Ueno H, Ogawa Y, Toguchi H. 【题名】:Pharmacokinetics of once-a-month injectable microspheres of leuprolide acetate. 【期刊】:Pharm Res. 【年、卷、期、起止页码】: 1991 Jun;8(6):787-91. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/1905810 【序号】:2 【作者】:Taguchi T1, Koyama H, Yayoi K, Wada T, Takatsuka Y, Sonoo H, Morimoto K, Tominaga T, Abe R, Enomoto K, et al. 【题名】:[Long-term clinical study on TAP-144-SR, an LH-RH agonist depot formulation, in premenopausal patients with advanced or recurrent breast cancer. TAP-144-SR Breast Cancer Study Group]. 【期刊】:Gan To Kagaku Ryoho. 【年、卷、期、起止页码】:1995 Mar;22(4):495-508. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/7887641 【序号】:3 【作者】:Niijima T1, Aso Y, Akaza H, Fujita K, Fuse H, Hosaka M, Isurugi K, Kamidono S, Katayama T, Kawabe K, et al. 【题名】:[Clinical phase I and phase II study on a sustained release formulation of leuprorelin acetate (TAP-144-SR), an LH-RH agonist, in patients with prostatic carcinoma. Collaborative++ Studies on Prostatic Carcinoma by the Study Group for TAP-144-SR]. 【期刊】:Hinyokika Kiyo. 【年、卷、期、起止页码】:1990 Nov;36(11):1343-60. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/2126912 【序号】:4 【作者】:D'Souza S1, Faraj JA, Dorati R, DeLuca PP. 【题名】:A short term quality control tool for biodegradable microspheres. 【期刊】:AAPS PharmSciTech. 【年、卷、期、起止页码】:2014 Jun;15(3):530-41. doi: 10.1208/s12249-013-0052-0. Epub 2014 Feb 12. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/24519488 【序号】:5 【作者】:Mashayekhi R1, Mobedi H, Najafi J, Enayati M. 【题名】:In-vitro/In-vivo comparison of leuprolide acetate release from an in-situ forming plga system. 【期刊】:Daru. 【年、卷、期、起止页码】:2013 Jul 15;21(1):57. doi: 10.1186/2008-2231-21-57. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/23856431 【序号】:6 【作者】:Schoubben A1, Blasi P, Deluca PP. 【题名】:Effect of agitation regimen on the in vitro release of leuprolide from poly(lactic-co-glycolic) acid microparticles. 【期刊】:J Pharm Sci. 【年、卷、期、起止页码】:2012 Mar;101(3):1212-20. doi: 10.1002/jps.23029. Epub 2011 Dec 21. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/22189694 【序号】:7 【作者】:D'Souza SS1, Faraj JA, DeLuca PP. 【题名】:A model-dependent approach to correlate accelerated with real-time release from biodegradable microspheres. 【期刊】:AAPS PharmSciTech. 【年、卷、期、起止页码】:2005 Oct 31;6(4):E553-64. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/16408857 【序号】:8 【作者】:D'Souza SS1, DeLuca PP. 【题名】:Development of a dialysis in vitro release method for biodegradable microspheres. 【期刊】:AAPS PharmSciTech. 【年、卷、期、起止页码】:2005 Oct 6;6(2):E323-8. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/16353991 【序号】:9 【作者】:Periti P1, Mazzei T, Mini E. 【题名】:Clinical pharmacokinetics of depot leuprorelin. 【期刊】:Clin Pharmacokinet. 【年、卷、期、起止页码】:2002;41(7):485-504. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/12083977 【序号】:10 【作者】:Shameem M1, Lee H, DeLuca PP. 【题名】:A short term (accelerated release) approach to evaluate peptide release from PLGA depot- formulations. 【期刊】:AAPS PharmSci. 【年、卷、期、起止页码】:1999;1(3):E7. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/11741203 【序号】:11 【作者】:Okada H1. 【题名】:One- and three-month release injectable microspheres of the LH-RH superagonist leuprorelin acetate. 【期刊】:Adv Drug Deliv Rev. 1 【年、卷、期、起止页码】:1997 Oct 13;28(1):43-70. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/10837564 【序号】:12 【作者】:Verspyck E1, Marpeau L, Lucas C. 【题名】:Leuprorelin depot 3.75 mg versus lynestrenol in the preoperative treatment of symptomatic uterine myomas: a multicentre randomised trial. 【期刊】:Eur J Obstet Gynecol Reprod Biol. 【年、卷、期、起止页码】:2000 Mar;89(1):7-13. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/10733017 【序号】:13 【作者】:Tunn UW1, Bargelloni U, Cosciani S, Fiaccavento G, Guazzieri S, Pagano F. 【题名】:Comparison of LH-RH analogue 1-month depot and 3-month depot by their hormone levels and pharmacokinetic profile in patients with advanced prostate cancer. 【期刊】:Urol Int. 【年、卷、期、起止页码】:1998;60 Suppl 1:9-16; discussion 16-7. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/9563139 【序号】:14 【作者】:Takada S1, Ogawa Y. 【题名】:. 【期刊】:Nihon Rinsho. 【年、卷、期、起止页码】:1998 Mar;56(3):675-9. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/9549355 【序号】:15 【作者】:Saruki K1, Sekihara T, Mashimo M, Matsuo H, Sekiguchi H. 【题名】:Leuprorelin acetate blood levels and dialysance after the administration of sustained-release leuprorelin acetate in a dialysis case complicated by prostate cancer. 【期刊】:Prostate. 【年、卷、期、起止页码】:1998 Feb 15;34(3):191-4. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/9492847 【序号】:16 【作者】:Okada H1, Doken Y, Ogawa Y, Toguchi H. 【题名】:Preparation of three-month depot injectable microspheres of leuprorelin acetate using biodegradable polymers. 【期刊】:Pharm Res. 【年、卷、期、起止页码】:1994 Aug;11(8):1143-7. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/7971715 【序号】:17 【作者】:Okada H1, Doken Y, Ogawa Y, Toguchi H. 【题名】:Sustained suppression of the pituitary-gonadal axis by leuprorelin three-month depot microspheres in rats and dogs. 【期刊】:Pharm Res. 【年、卷、期、起止页码】:1994 Aug;11(8):1199-203. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/7971724 【序号】:18 【作者】:Toguchi H1. 【题名】:Formulation study of leuprorelin acetate to improve clinical performance. 【期刊】:Clin Ther. 【年、卷、期、起止页码】:1992;14 Suppl A:121-30. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/1606592 【序号】:19 【作者】:Asano M1, Fukuzaki H, Yoshida M, Kumakura M, Mashimo T, Yuasa H, Imai K, Yamanaka H. 【题名】:In vivo characteristics of low molecular weight copoly (D,L-lactic acid) formulations with controlled release of LH-RH agonist. 【期刊】:Biomaterials. 【年、卷、期、起止页码】:1989 Oct;10(8):569-73. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/2513891 【序号】:20 【作者】:Ogawa Y1, Okada H, Heya T, Shimamoto T. 【题名】:Controlled release of LHRH agonist, leuprolide acetate, from microcapsules: serum drug level profiles and pharmacological effects in animals. 【期刊】:J Pharm Pharmacol. 【年、卷、期、起止页码】:J Pharm Pharmacol. 1989 Jul;41(7):439-44. 【全文链接】:https://www.ncbi.nlm.nih.gov/pubmed/2570847