speleers
第1楼2008/09/26
目录:
1 Overview Drug Metabolism in the Modern Pharmaceutical Industry
2 Oxidative, Reductive, and Hydrolytic Metabolism of Drugs
3 Conjugative Metabolism of Drugs
4 Enzyme Kinetics
5 Metabolism-Mediated Drug-Drug Interactions
6 Drug Transporters in Drug Disposition, Drug Interactions, and Drug Resistance
7 Regulatory Considerations of Drug Metabolism and Drug Interaction Studies
8 Drug Metabolism Research as an Integral Part of the Drug Discovery Process
9 Role of Drug Metabolism in Drug Development
10 Applications of Liquid Radiochromatography Techniques in Drug Metabolism Studies
11 Application of Liquid Chromatography Mass Spectrometry for Metabolite Identification
12 Introduction to NMR and Its Application in Metabolite Structure Determination
13 Determination of Metabolic Rates and Enzyme Kinetics
14 Protocols for Assessment of In vitro and In vivo Bioactivation Potential of Drug Candidates
15 Reaction Phenotyping
16 Analysis of In vitro Cytochrome P450 Inhibition in Drug Discovery and Development
17 Testing Drug Candidates for CYP3A4 Induction
18 ADME Studies in Animals and Humans Experimental Design, Metabolite Profiling and Identification, and Data Presentation
rwc5654105
第6楼2008/11/07
太谢谢了!刚好是我感兴趣的专业,终于能证明药物代谢动力学在新药研发中的极其重要地位了!