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【资料】Drug Metabolism in Drug Design and Development

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  • 该帖子已被版主-jiangkezhi加2积分,加2经验;加分理由:积极提供质谱应用相关资料
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  • speleers

    第1楼2008/09/26

    目录:
    1 Overview Drug Metabolism in the Modern Pharmaceutical Industry
    2 Oxidative, Reductive, and Hydrolytic Metabolism of Drugs
    3 Conjugative Metabolism of Drugs
    4 Enzyme Kinetics
    5 Metabolism-Mediated Drug-Drug Interactions
    6 Drug Transporters in Drug Disposition, Drug Interactions, and Drug Resistance
    7 Regulatory Considerations of Drug Metabolism and Drug Interaction Studies
    8 Drug Metabolism Research as an Integral Part of the Drug Discovery Process
    9 Role of Drug Metabolism in Drug Development
    10 Applications of Liquid Radiochromatography Techniques in Drug Metabolism Studies
    11 Application of Liquid Chromatography Mass Spectrometry for Metabolite Identification
    12 Introduction to NMR and Its Application in Metabolite Structure Determination
    13 Determination of Metabolic Rates and Enzyme Kinetics
    14 Protocols for Assessment of In vitro and In vivo Bioactivation Potential of Drug Candidates
    15 Reaction Phenotyping
    16 Analysis of In vitro Cytochrome P450 Inhibition in Drug Discovery and Development
    17 Testing Drug Candidates for CYP3A4 Induction
    18 ADME Studies in Animals and Humans Experimental Design, Metabolite Profiling and Identification, and Data Presentation

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  • xiao201

    第2楼2008/09/26

    多谢多谢,一定认真学习

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  • uu325

    第3楼2008/10/08

    太谢谢LZ了,我们体内药分老师极力推荐这本书呢!!

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  • 天字一号猪

    第7楼2008/11/07

    应助达人

    不懂,但是顶一下!

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  • yuduoling

    第8楼2008/11/10

    学习中,多谢分享

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  • basin_1982

    第9楼2009/06/18

    真是好东西,谢谢了。

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  • caicaiseven

    第10楼2009/07/15

    太感谢楼主了!!! 正在找这本书啊~~~

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